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Drug Name EPZ015666
Trade Name
Synonyms GSK3235025
Drug Descriptions

EPZ015666 (GSK3235025) selectively inhibits protein arginine methyltransferase-5 (PRMT5), which may lead to anti-tumor activity (PMID: 25915199, PMID: 31694585).

DrugClasses PRMT5 Inhibitor 12
CAS Registry Number 1616391-65-1


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Therapy Name Drugs Efficacy Evidence Clinical Trials
EPZ015666 EPZ015666 0 0
EPZ015666 + MS023 EPZ015666 MS023 0 0

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