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Drug Name TAS0612
Trade Name
Synonyms TAS-0612|TAS 0612
Drug Descriptions

TAS0612 is a multikinase inhibitor that blocks the activity of Akt, p70S6K, and p90RSK, and decreases phosphorylation of Ybx1, potentially resulting in reduced tumor cell proliferation and inhibition of tumor growth (PMID: 31879363).

DrugClasses Akt Inhibitor (Pan) 21
CAS Registry Number NA
NCIT ID C175557

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Therapy Name Drugs Efficacy Evidence Clinical Trials
Futibatinib + TAS0612 Futibatinib TAS0612 0 0
TAS0612 TAS0612 4 1


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