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Drug Name | Fenebrutinib |
Trade Name | |
Synonyms | GDC-0853 |
Drug Descriptions |
Fenebrutinib (GDC-0853) is a small molecule inhibitor of BTK, including BTK C481S, which may result in reduced BTK activity, increased cytotoxicity, and antitumor activity (PMID: 30018078, PMID: 29560128). |
DrugClasses | BTK inhibitor 36 |
CAS Registry Number | 1434048-34-6 |
NCIT ID | C116844 |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
Fenebrutinib | Fenebrutinib | 0 | 0 |