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Drug Name BLU-701
Trade Name
Synonyms BLU701|BLU 701
Drug Descriptions

BLU-701 is a reversible EGFR inhibitor that blocks the activity of mutant forms of EGFR, including C797S, while sparing wild-type EGFR, which results in reduced downstream signaling and potentially leads to decreased tumor growth (Cancer Res 2021;81(13_Suppl):Abstract nr 1262).

DrugClasses EGFR Inhibitor 4th gen 7
CAS Registry Number NA
NCIT ID C185863


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Therapy Name Drugs Efficacy Evidence Clinical Trials
BLU-701 BLU-701 0 1
BLU-701 + Carboplatin + Pemetrexed Disodium BLU-701 Carboplatin Pemetrexed Disodium 0 1
BLU-701 + Osimertinib BLU-701 Osimertinib 0 1

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