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Drug Name APS03118
Trade Name APS 03118|APS-03118
Drug Descriptions

APS03118 is a RET inhibitor with activity against RET fusions and gatekeeper mutations, potentially inhibiting phosphorylation, proliferation, and tumor growth (J Clin Oncol 40, no. 16_suppl (June 1, 2022)).

DrugClasses RET Inhibitor 48
CAS Registry Number NA


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Therapy Name Drugs Efficacy Evidence Clinical Trials
APS03118 APS03118 8 0

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