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Drug Name | Bafetinib |
Trade Name | |
Synonyms | NS-187|INNO-406 |
Drug Descriptions |
Bafetinib (NS-187) is a tyrosine kinase inhibitor with activity against Lyn, SRC kinase, DDR1/2, and BCR-ABL, but not the T315I mutation (PMID: 21154127, PMID: 19890374). |
DrugClasses | BCR-ABL Inhibitor 31 DDR1 Inhibitor 10 DDR2 inhibitor 7 LYN Inhibitor 3 |
CAS Registry Number | 859212-16-1 |
NCIT ID | C62516 |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
Bafetinib | Bafetinib | 0 | 0 |