Drug Detail


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Drug Name BMS-754807
Trade Name
Drug Descriptions

BMS-754807 is a multi-kinase inhibitor with activity against IGF-1R, insulin receptor, MET, ALK, TRKA, TRKB, AURKA, and AURKB, potentially resulting in decreased tumor cell proliferation (PMID: 25748921, PMID: 31433065).

DrugClasses ALK Inhibitor 32 Aurka Inhibitors 27 Aurkb Inhibitors 21 IGF-1R Inhibitor 17 MET Inhibitor 59 TrkA Receptor Inhibitor 8
CAS Registry Number 1001350-96-4
NCIT ID C74043


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Therapy Name Drugs Efficacy Evidence Clinical Trials
AZD8055 + BMS-754807 AZD8055 BMS-754807 0 0
BMS-754807 BMS-754807 0 0
BMS-754807 + Dacomitinib BMS-754807 Dacomitinib 0 0
BMS-754807 + Everolimus BMS-754807 Everolimus 0 0
BMS-754807 + Midostaurin BMS-754807 Midostaurin 0 0
BMS-754807 + SCH772984 BMS-754807 SCH772984 0 0

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