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Drug Name CI-1040
Trade Name
Synonyms PD184352|PD-184352
Drug Descriptions

CI-1040 (PD184352) binds and inhibits Mek1 and Mek2, which may inhibit the activation of downstream signaling targets and reduce tumor cell proliferation (PMID: 14613031, PMID: 16009947).

DrugClasses MEK inhibitor (Pan) 22 MEK1 Inhibitor 20 MEK2 Inhibitor 18

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Therapy Name Drugs Efficacy Evidence Clinical Trials
CI-1040 CI-1040 16 0
CI-1040 + WZ4002 CI-1040 WZ4002 0 0


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