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Drug Name | CUDC-101 |
Trade Name | |
Synonyms | |
Drug Descriptions |
CUDC-101 is a small-molecule inhibitor of EGFR, ERBB2 (HER2), and class I and II HDACs, which has demonstrated activity in EGFR-inhibitor resistant tumor cell lines (PMID: 20388807, PMID: 23536719, PMID: 31584454). |
DrugClasses | EGFR Inhibitor (Pan) 61 HDAC Inhibitor 45 HER2 Inhibitor 41 |
CAS Registry Number | 1012054-59-9 |
NCIT ID | C78850 |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
CUDC-101 | CUDC-101 | 0 | 0 |