Drug Detail

Contact

Missing content? – Request curation!

Request curation for specific Genes, variants, or PubMed publications.

Have questions, comments or suggestions? - Let us know!

Email us at : ckbsupport@jax.org

Drug Name Taselisib
Trade Name
Synonyms RG7606|GDC-0032
Drug Descriptions

Taselisib (GDC-0032) is a beta isoform-sparing PI3K inhibitor, with greater activity against oncogenic mutants of PIK3CA (PMID: 23662903).

DrugClasses PIK3CA inhibitor 16 PIK3CD inhibitor 25 PIK3CG inhibitor 8

Filtering

  • Case insensitive filtering will display rows where any text in any cell matches the filter term
  • Simple literal full or partial string matches
  • Separate multiple filter terms with a spaces, order doesn't matter (a b c and c b a are equivalent )
  • Filtering will only apply to rows that are already loaded on the page, filtering has no impact on query parameters
  • Use quotes to match a longer phrase which contains spaces "mtor c1483f"

Sorting

  • Generally, the default sort order for tables is set to be first column ascending, however, specific tables may set a different default sort order.
  • Click on any column header arrows to sort by that column
  • Hold down the Shift key and click multiple columns to sort by more than one column, be sure to set ascending or descending order for a given column, before moving on to the next column.

Therapy Name Drugs Efficacy Evidence Clinical Trials
Docetaxel + Taselisib Docetaxel Taselisib 0 1
Enzalutamide + Taselisib Enzalutamide Taselisib 0 1
Fulvestrant + Taselisib Fulvestrant Taselisib 0 0
Letrozole + Taselisib Letrozole Taselisib 1 0
Neratinib + Taselisib Neratinib Taselisib 3 0
Paclitaxel + Taselisib Paclitaxel Taselisib 0 1
Radiotherapy + Taselisib Radiotherapy Taselisib 3 0
Tamoxifen + Taselisib Tamoxifen Taselisib 0 0
Taselisib Taselisib 17 7


Additional content available in CKB BOOST