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Drug Name Sapanisertib
Trade Name
Synonyms INK128|INK-128|TAK-228|MLN0128|MLN-0128
Drug Descriptions

Sapanisertib (MLN0128) is an ATP-competitive mTOR kinase inhibitor that induces apoptosis and inhibits growth in tumor cells (PMID: 25519700, PMID: 32488989).

DrugClasses mTOR Inhibitor 51
CAS Registry Number 224844-38-5
NCIT ID C90548

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Therapy Name Drugs Efficacy Evidence Clinical Trials
ABT-737 + Sapanisertib ABT-737 Sapanisertib 1 0
Ado-trastuzumab emtansine + Sapanisertib Ado-trastuzumab emtansine Sapanisertib 0 0
Aflibercept + Sapanisertib Aflibercept Sapanisertib 0 1
Alisertib + Sapanisertib Alisertib Sapanisertib 0 2
AZD4547 + Sapanisertib AZD4547 Sapanisertib 0 0
Bevacizumab + Sapanisertib Bevacizumab Sapanisertib 0 1
Carboplatin + Paclitaxel + Sapanisertib Carboplatin Paclitaxel Sapanisertib 1 1
EHop-016 + Sapanisertib EHop-016 Sapanisertib 0 0
Erdafitinib + Sapanisertib Erdafitinib Sapanisertib 0 0
Exemestane + Sapanisertib Exemestane Sapanisertib 0 1
Fulvestrant + Sapanisertib Fulvestrant Sapanisertib 0 2
Ibrutinib + Sapanisertib Ibrutinib Sapanisertib 0 0
Infigratinib + Sapanisertib Infigratinib Sapanisertib 0 0
Linsitinib + Sapanisertib Linsitinib Sapanisertib 0 0
Linsitinib + Sapanisertib + Trametinib Linsitinib Sapanisertib Trametinib 0 0
Metformin + Sapanisertib Metformin Sapanisertib 0 1
Mobocertinib + Sapanisertib Mobocertinib Sapanisertib 0 0
Neratinib + Sapanisertib Neratinib Sapanisertib 0 0
Osimertinib + Sapanisertib Osimertinib Sapanisertib 0 2
Paclitaxel + Sapanisertib + Serabelisib Paclitaxel Sapanisertib Serabelisib 0 1
PD-0325901 + Sapanisertib PD-0325901 Sapanisertib 4 0
Phenformin + Sapanisertib Phenformin Sapanisertib 0 0
Ponatinib + Sapanisertib Ponatinib Sapanisertib 0 0
Sapanisertib Sapanisertib 6 19
Sapanisertib + SBI-0206965 SBI-0206965 Sapanisertib 0 0
Sapanisertib + Serabelisib Sapanisertib Serabelisib 0 4
Sapanisertib + Sirolimus Sapanisertib Sirolimus 0 0
Sapanisertib + Tamoxifen Sapanisertib Tamoxifen 0 1
Sapanisertib + Telaglenastat Sapanisertib Telaglenastat 0 1
Sapanisertib + Tipifarnib Sapanisertib Tipifarnib 1 0
Sapanisertib + Tovorafenib Sapanisertib Tovorafenib 0 1
Sapanisertib + Trametinib Sapanisertib Trametinib 0 0
Sapanisertib + WEHI-539 Sapanisertib WEHI-539 1 0


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