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Drug Name AMG 458
Trade Name
Synonyms AMG-458|AMG458
Drug Descriptions

AMG 458 inhibits wild-type and mutant forms of MET and has additional activity against MST1R (RON), resulting in decreased tumor growth (PMID: 20015007, PMID: 22836051).

DrugClasses MET Inhibitor 59 RON Inhibitor 11
CAS Registry Number 913376-83-7
NCIT ID NA

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Therapy Name Drugs Efficacy Evidence Clinical Trials
AMG 458 AMG 458 0 0


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