Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@jax.org
Drug Name | Semagacestat |
Trade Name | |
Synonyms | LY450139|LY-450139 |
Drug Descriptions |
Semagacestat (LY450139) is a gamma secretase inhibitor, which blocks Notch cleavage and activation, and may inhibit angiogenesis and tumor growth (PMID: 22323718, PMID: 28978478). |
DrugClasses | Gamma secretase inhibitor 13 |
CAS Registry Number | 425386-60-3 |
NCIT ID | C81115 |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
Semagacestat | Semagacestat | 0 | 0 |