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Drug Name Z-endoxifen HCl
Trade Name
Synonyms Endoxifen Hydrochloride
Drug Descriptions

Z-endoxifen HCl is the active metabolite of tamoxifen, which competitively inhibits estradiol binding to estrogen receptors (ER), thereby inhibiting growth of ER-positive tumors (PMID: 26232141).

DrugClasses Hormone Antineoplastics 5
CAS Registry Number 1032008-74-4
NCIT ID C95713


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Therapy Name Drugs Efficacy Evidence Clinical Trials
Goserelin + Z-endoxifen HCl Goserelin Z-endoxifen HCl 0 1
Z-endoxifen HCl Z-endoxifen HCl 0 3

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