Drug Detail


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Drug Name MK8033
Trade Name
Synonyms MK-8033|HQP8361|HQP 8361|HQP-8361|MK 8033
Drug Descriptions

MK8033 is an inhibitor of MET and MST1R (RON) that suppresses mTOR signaling, potentially resulting in reduced survival and colony formation, increased apoptosis, and inhibition of tumor growth (PMID: 23792360, PMID: 33163272).

DrugClasses MET Inhibitor 58 RON Inhibitor 11
CAS Registry Number 1196681-38-5
NCIT ID C116866


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Therapy Name Drugs Efficacy Evidence Clinical Trials
MK8033 MK8033 0 0
MK8033 + Osimertinib MK8033 Osimertinib 0 0

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