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Drug Name PF-3758309
Trade Name
Synonyms
Drug Descriptions

PF-3758309 is a p21-activated kinase (PAK) inhibitor with activity against PAK1 and PAK4, potentially resulting in decreased tumor growth (PMID: 20439741, PMID: 23543898, PMID: 32469945, PMID: 31312349).

DrugClasses Pak-I Inhibitor 4

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Therapy Name Drugs Efficacy Evidence Clinical Trials
JQ1 + PF-3758309 JQ1 PF-3758309 0 0
PF-3758309 PF-3758309 0 0


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