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Drug Name FRAX1036
Trade Name
Synonyms FRAX-1036
Drug Descriptions

FRAX1036 is an inhibitor of group I PAKs (PAK1, PAK2, and PAK3), which may result in increased tumor cell apoptosis and sensitivity to microtubule-targeted agents (PMID: 25902869).

DrugClasses PAK1 Inhibitor 11
CAS Registry Number 1432908-05-8
NCIT ID NA

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Therapy Name Drugs Efficacy Evidence Clinical Trials
BDP9066 + FRAX1036 BDP9066 FRAX1036 0 0
Docetaxel + FRAX1036 Docetaxel FRAX1036 0 0
Everolimus + FRAX1036 Everolimus FRAX1036 0 0
FRAX1036 FRAX1036 0 0
FRAX1036 + Lenvatinib FRAX1036 Lenvatinib 0 0


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