Drug Detail

Drug Name GS-5829
Trade Name
Drug Descriptions

GS-5829 is a BET bromodomain inhibitor, potentially resulting in inhibition of cell growth and apoptotic activity (Blood 2016 128:5104).

DrugClasses BET Inhibitor (Pan) 25


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Therapy Name Drugs Efficacy Evidence Clinical Trials
Exemestane + GS-5829 Exemestane GS-5829 0 3
Fulvestrant + GS-5829 Fulvestrant GS-5829 0 1
GS-5829 GS-5829 0 0
GS-5829 + Venetoclax GS-5829 Venetoclax 2 0

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