Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@jax.org
Drug Name | RVX-208 |
Trade Name | |
Synonyms | Apabetalone |
Drug Descriptions |
Apabetalone (RVX-208) is a bromo and extraterminal (BET) protein inhibitor that selectively binds to the second bromodomain found on BET proteins, resulting in inhibition of downstream gene transcription (PMID: 24248379, PMID: 31257080). |
DrugClasses | BET Inhibitor (Pan) 32 |
CAS Registry Number | 1044870-39-4 |
NCIT ID | C171748 |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
RVX-208 | RVX-208 | 0 | 0 |