Drug Detail


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Drug Name CPI-455
Trade Name
Drug Descriptions

CPI-455 is an inhibitor of KDM5A, KDM5B, and KDM5C, which may reduce cell survival, in particular those cells that are considered drug resistant (PMID: 27214401, PMID: 31238504).

CAS Registry Number NA


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Therapy Name Drugs Efficacy Evidence Clinical Trials
AZ628 + CPI-455 AZ628 CPI-455 0 0
CPI-455 CPI-455 0 0
CPI-455 + Erlotinib CPI-455 Erlotinib 0 0
CPI-455 + Lapatinib CPI-455 Lapatinib 0 0
CPI-455 + Vemurafenib CPI-455 Vemurafenib 0 0

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