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Drug Name | GDC-0077 |
Trade Name | |
Synonyms | RO7113755|RG6114|GDC0077|GDC 0077|inavolisib |
Drug Descriptions |
GDC-0077 inhibits PIK3CA, with selectivity for mutant PIK3CA over wild-type PIK3CA, potentially resulting in increased apoptosis and decreased growth of PIK3CA-mutant tumors (AACR; Cancer Res 2017;77(13 Suppl):Abstract nr 156). |
DrugClasses | PIK3CA inhibitor 21 |
CAS Registry Number | 2060571-02-8 |
NCIT ID | C132166 |