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Drug Name | Inavolisib |
Trade Name | |
Synonyms | GDC-0077|RO7113755|RG6114|GDC0077|GDC 0077 |
Drug Descriptions |
Inavolisib (GDC-0077) inhibits PIK3CA, with selectivity for mutant PIK3CA over wild-type PIK3CA, potentially resulting in increased apoptosis and decreased growth of PIK3CA-mutant tumors (PMID: 36455032). |
DrugClasses | PIK3CA inhibitor 23 |
CAS Registry Number | 2060571-02-8 |
NCIT ID | C132166 |