Drug Detail


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Drug Name EED226
Trade Name
Drug Descriptions

EED226 is a small molecule inhibitor of PRC2 via direct binding to the H3K27me3 pocket of EED, which leads to altered PRC2 targeted gene expression and thus, may result in inhibition of cell proliferation, blockade of tumor growth, and tumor regression (PMID: 28135235).

CAS Registry Number NA


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Therapy Name Drugs Efficacy Evidence Clinical Trials
EED226 EED226 0 0
EED226 + EI1 EED226 EI1 0 0
EED226 + Pomalidomide EED226 Pomalidomide 0 0

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