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Drug Name CEP-11981
Trade Name
Synonyms ESK981|CEP11981|CEP 11981
Drug Descriptions

CEP-11981 is a multikinase inhibitor that targets VEGFR1-3 and TIE2, which may inhibit tumor angiogenesis and lead to tumor growth inhibition (PMID: 24982343, PMID: 25152243).

DrugClasses TIE2 Inhibitor 3 VEGFR Inhibitor (Pan) 33
CAS Registry Number 856691-93-5
NCIT ID C82379

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Therapy Name Drugs Efficacy Evidence Clinical Trials
CEP-11981 CEP-11981 0 2
CEP-11981 + Nivolumab CEP-11981 Nivolumab 0 2


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