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Drug Name Bozitinib
Trade Name
Synonyms PLB1001|PLB-1001|APL-101|APL 101|APL101
Drug Descriptions

Bozitinib (PLB-1001) is an ATP-competitive, small molecule inhibitor of MET, which is able to permeate the blood brain barrier and may inhibit downstream signaling and block tumor growth (PMID: 30343896).

DrugClasses MET Inhibitor 54
CAS Registry Number 1440964-89-5
NCIT ID C129717

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Therapy Name Drugs Efficacy Evidence Clinical Trials
Bozitinib Bozitinib 0 1
Bozitinib + Osimertinib Bozitinib Osimertinib 0 1


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