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Drug Name MA242
Trade Name
Synonyms MA 242|MA-242
Drug Descriptions

MA242 binds to and inhibits MDM2 and NFAT1, leading to ubiquitination and degradation of MDM2, which may lead to apoptosis and inhibition of tumor cell growth and metastasis independent of Tp53 function (PMID: 30217928).

DrugClasses MDM2 Inhibitor 19

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Therapy Name Drugs Efficacy Evidence Clinical Trials
Gemcitabine + MA242 Gemcitabine MA242 0 0
MA242 MA242 0 0


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