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Drug Name GSK2801
Trade Name
Synonyms GSK 2801|GSK-2801
Drug Descriptions

GSK2801 is a bromodomain inhibitor that selectively inhibits BAZ2A/B and BRD9, which has potential antitumor activity (PMID: 31000582).

DrugClasses
CAS Registry Number 1619994-68-1
NCIT ID NA

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Therapy Name Drugs Efficacy Evidence Clinical Trials
Birabresib + GSK2801 Birabresib GSK2801 0 0
GSK2801 GSK2801 0 0
GSK2801 + HY-16462 GSK2801 HY-16462 0 0
GSK2801 + JQ1 GSK2801 JQ1 0 0


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