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Therapy Name GLPG0187
Synonyms
Therapy Description

GLPG0187 is an integrin receptor antagonist, which may decrease angiogenesis and reduce tumor growth and metastasis (PMID: 25156971, PMID: 26792581).

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Drug Name Trade Name Synonyms Drug Classes Drug Description
GLPG0187 GLPG0187 is an integrin receptor antagonist, which may decrease angiogenesis and reduce tumor growth and metastasis (PMID: 25156971, PMID: 26792581).

Filtering

  • Case insensitive filtering will display rows where any text in any cell matches the filter term
  • Simple literal full or partial string matches
  • Separate multiple filter terms with a spaces, order doesn't matter (a b c and c b a are equivalent )
  • Filtering will only apply to rows that are already loaded on the page, filtering has no impact on query parameters
  • Use quotes to match a longer phrase which contains spaces "mtor c1483f"

Sorting

  • Generally, the default sort order for tables is set to be first column ascending, however, specific tables may set a different default sort order.
  • Click on any column header arrows to sort by that column
  • Hold down the Shift key and click multiple columns to sort by more than one column, be sure to set ascending or descending order for a given column, before moving on to the next column.

Molecular Profile Indication/Tumor Type Response Type Therapy Name Approval Status Evidence Type Efficacy Evidence References
Unknown unknown Advanced Solid Tumor no benefit GLPG0187 Phase I Actionable In a Phase I trial, continuous treatment with GLPG0187 demonstrated safety but lack of efficacy, with 15% (3/20) of patients demonstrating stable disease and no patients with tumor response (PMID: 26792581). 26792581

Filtering

  • Case insensitive filtering will display rows where any text in any cell matches the filter term
  • Simple literal full or partial string matches
  • Separate multiple filter terms with a spaces, order doesn't matter (a b c and c b a are equivalent )
  • Filtering will only apply to rows that are already loaded on the page, filtering has no impact on query parameters
  • Use quotes to match a longer phrase which contains spaces "mtor c1483f"

Sorting

  • Generally, the default sort order for tables is set to be first column ascending, however, specific tables may set a different default sort order.
  • Click on any column header arrows to sort by that column
  • Hold down the Shift key and click multiple columns to sort by more than one column, be sure to set ascending or descending order for a given column, before moving on to the next column.

Clinical Trial Phase Therapies Title Recruitment Status


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