Drug Detail


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Drug Name RLY-4008
Trade Name
Synonyms RLY4008|RLY 4008
Drug Descriptions

RLY-4008 binds to and inhibits FGFR2, selectively targeting primary oncogenic FGFR2 mutations and leads to decreased FGFR2-dependent signaling, potentially resulting in inhibition of tumor cell proliferation (NCI Drug Dictionary; Journal of Clinical Oncology 39, no. 15_suppl).

DrugClasses FGFR2 Inhibitor 19
CAS Registry Number NA
NCIT ID C174208


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Therapy Name Drugs Efficacy Evidence Clinical Trials
RLY-4008 RLY-4008 6 1

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