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Drug Name JAB-8263
Trade Name
Synonyms JAB8263|JAB 8263
Drug Descriptions

JAB-8263 is a BET inhibitor that that binds BRD2, BRD3, BRD4, and BRDT and prevents their interaction with acetylated histones, thereby leading to altered chromatin modeling and gene expression patterns, and potentially resulting in inhibition of tumor cell growth (NCI Drug Dictionary).

DrugClasses BET Inhibitor (Pan) 32
CAS Registry Number NA
NCIT ID C179628

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Therapy Name Drugs Efficacy Evidence Clinical Trials
JAB-8263 JAB-8263 0 1


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