Drug Detail


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Drug Name KT-253
Trade Name
Synonyms KT 253|KT253
Drug Descriptions

KT-253 is a degrader of MDM2, which reduces TP53-dependent increase in MDM2 protein levels and potentially induces apoptosis in tumor cells and inhibits tumor growth (Blood (2022) 140 (Supplement 1): 6239-6240).

DrugClasses MDM2 Inhibitor 22
CAS Registry Number NA


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Therapy Name Drugs Efficacy Evidence Clinical Trials
KT-253 KT-253 0 1

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