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Drug Name | Staurosporine |
Trade Name | |
Synonyms | CGP-39360|AM-2282 |
Drug Descriptions |
Staurosporine (CGP-39360) is an alkaloid pan-protein kinase C (PKC) inhibitor, with activity against several additional protein kinases, including PAK1 (PMID: 32863957), which may result in increased apoptosis and decreased tumor cell growth (PMID: 3457562, PMID: 8529658, PMID: 8913270). |
DrugClasses | PAK1 Inhibitor 11 PKC Inhibitor (Pan) 11 |
CAS Registry Number | 62996-74-1 |
NCIT ID | C1237 |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
Staurosporine | Staurosporine | 0 | 0 |