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Drug Name | K252a |
Trade Name | |
Synonyms | K252-a|K252 a|K-252a |
Drug Descriptions |
K-252a is an ATP-competitive inhibitor of cyclic nucleotide-dependent protein kinases and protein kinase C, and also has inhibitory activity againstTRKs and MET, potentially resulting in decreased downstream signaling and reduced tumor cell proliferation (PMID: 3028414, PMID: 12118367). |
DrugClasses | MET Inhibitor 59 PKC Inhibitor (Pan) 11 Trk Receptor Inhibitor (Pan) 31 |
CAS Registry Number | 99533-80-9 |
NCIT ID | C1382 |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
K252a | K252a | 0 | 0 |