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Drug Name | SU11652 |
Trade Name | |
Synonyms | SU-11652 |
Drug Descriptions |
SU11652 is an inhibitor of multiple tyrosine kinase receptors including Pdgfr-beta, Kdr (Vegfr2), Fgfr1, and Kit, which blocks pathway activation, promotes cell cycle arrest, and induces apoptosis of tumor cells (PMID: 12091352, PMID: 23216927). |
DrugClasses | FGFR1 Inhibitor 28 KIT Inhibitor 57 PDGFR-beta Inhibitor 14 VEGFR2 Inhibitor 37 |
CAS Registry Number | 326914-10-7 |
NCIT ID | NA |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
SU11652 | SU11652 | 0 | 0 |