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Drug Name | GSK503 |
Trade Name | |
Synonyms | GSK-503|GSK 503 |
Drug Descriptions |
GSK503 selectively inhibits EZH2, resulting in decreased EZH2 methytransferase activity, and potentially leading to reduced tumor growth (PMID: 23680150, PMID: 28228601, PMID: 29732557). |
DrugClasses | EZH2 inhibitor 20 |
CAS Registry Number | 1346572-63-1 |
NCIT ID | NA |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
GSK503 | GSK503 | 0 | 0 |