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Drug Name GS716054
Trade Name
Synonyms
Drug Descriptions

GS716054 inhibits KDM5, which increases H3K4 tri-methylation and potentially induces cell cycle arrest and decreases proliferation of tumor cells (PMID: 38351059).

DrugClasses
CAS Registry Number NA
NCIT ID NA

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Therapy Name Drugs Efficacy Evidence Clinical Trials
GS716054 GS716054 0 0
GS716054 + Ibrutinib GS716054 Ibrutinib 0 0


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