Drug Detail


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Drug Name GSK461364
Trade Name
Drug Descriptions

GSK461364 is a specific ATP-competitive inhibitor of PLK1 that induces mitotic arrest, leading to cell death in many cancer cell lines (PMID: 19474163, PMID: 31751384).

DrugClasses PLK1 Inhibitor 18
CAS Registry Number 929095-18-1
NCIT ID C70948


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Therapy Name Drugs Efficacy Evidence Clinical Trials
GSK461364 GSK461364 0 0
GSK461364 + Palbociclib GSK461364 Palbociclib 1 0

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