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Drug Name CCT241533
Trade Name
Synonyms CCT 241533|CCT-241533
Drug Descriptions

CCT241533 is an ATP-competitive inhibitor of CHK2, which enhances PARP inhibitor efficacy in cells lacking functional TP53 (PMID: 21239475).

DrugClasses CHK2 Inhibitor 7
CAS Registry Number 1262849-73-9


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Therapy Name Drugs Efficacy Evidence Clinical Trials
CCT241533 CCT241533 0 0
CCT241533 + Olaparib CCT241533 Olaparib 0 0
CCT241533 + Rucaparib CCT241533 Rucaparib 0 0

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