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Drug Name BPTES
Trade Name
Synonyms bis-2-(5-phenylacetamido-1,2,4-thiadiazol-2-yl)ethyl sulfide
Drug Descriptions

BPTES is a small molecule that inhibits glutaminase, which results in decreased conversion of glutamine to glutamate, and potentially leads to decreased tumor cell growth (PMID: 21045145, PMID: 25915584, PMID: 32450839).

DrugClasses Glutaminase Inhibitor 3
CAS Registry Number 314045-39-1
NCIT ID NA

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Therapy Name Drugs Efficacy Evidence Clinical Trials
BPTES BPTES 2 0
BPTES + Olaparib BPTES Olaparib 1 0


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