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Drug Name | GNE-272 |
Trade Name | |
Synonyms | |
Drug Descriptions |
GNE-272 is an inhibitor targeting the bromodomains of CREBBP and EP300, which subsequently prevents MYC expression, thereby potentially resulting in anti-proliferative effects and tumor growth inhibition (PMID: 27682507). |
DrugClasses | CBP/p300 inhibitor 11 |
CAS Registry Number | 1936428-93-1 |
NCIT ID | NA |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
GNE-272 | GNE-272 | 0 | 0 |