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Drug Name ARV-771
Trade Name
Synonyms ARV 771|ARV771
Drug Descriptions

ARV-771 is a bifunctional molecule that targets BET proteins for proteolytic degradation, resulting in reduced target gene expression and potentially leading to increased apoptosis and reduced tumor growth (PMID: 31217338, PMID: 27274052, PMID: 30575820).

DrugClasses BET Inhibitor (Pan) 32
CAS Registry Number 1949837-12-0
NCIT ID NA

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Therapy Name Drugs Efficacy Evidence Clinical Trials
ARV-771 ARV-771 0 0
ARV-771 + Enzastaurin ARV-771 Enzastaurin 0 0


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