Drug Detail


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Drug Name EPI-7386
Trade Name
Synonyms EPI7386|EPI 7386
Drug Descriptions

EPI-7386 is an N-terminal domain AR inhibitor that blocks transcriptional activity of both full-length and splice variants of AR, potentially leading to antitumor effects (Mol Cancer Ther 2019;18(12 Suppl):Abstract nr B117).

DrugClasses Hormone - Anti-androgens 47
CAS Registry Number NA
NCIT ID C173374


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Therapy Name Drugs Efficacy Evidence Clinical Trials
Abiraterone + EPI-7386 + Prednisone Abiraterone EPI-7386 Prednisone 0 1
Apalutamide + EPI-7386 Apalutamide EPI-7386 0 1
Enzalutamide + EPI-7386 EPI-7386 Enzalutamide 0 1
EPI-7386 EPI-7386 0 1

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