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| Drug Name | Enzalutamide |
| Trade Name | Xtandi |
| Synonyms | MDV3100|ASP9785 |
| Drug Descriptions |
Xtandi (enzalutamide) is a second-generation small molecule androgen receptor (AR) inhibitor that inhibits AR signaling, thereby resulting in decreased tumor growth (PMID: 24009414, PMID: 25945058). Xtandi (enzalutamide) is FDA approved for use in patients with castration-resistant prostate cancer and metastatic hormone-sensitive prostate cancer (FDA.gov). |
| DrugClasses | Hormone - Anti-androgens 41 |
| CAS Registry Number | 915087-33-1 |
| NCIT ID | C71744 |
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