Drug Detail

Contact

Missing content? – Request curation!

Request curation for specific Genes, variants, or PubMed publications.

Have questions, comments or suggestions? - Let us know!

Email us at : ckbsupport@jax.org

Drug Name Relugolix
Trade Name
Synonyms TAK-385|Relumina
Drug Descriptions

Relugolix (TAK-385) is a gonadotropin-releasing hormone antagonist, which binds to the gonadotropin-releasing hormone receptor, thereby preventing the secretion and release of luteinizing hormone and follicle stimulating hormone and possibly resulting in anti-tumor activity (PMID: 32469183).

DrugClasses
CAS Registry Number 737789-87-6
NCIT ID C114498

Filtering

  • Case insensitive filtering will display rows where any text in any cell matches the filter term
  • Simple literal full or partial string matches
  • Separate multiple filter terms with a spaces, order doesn't matter (a b c and c b a are equivalent )
  • Filtering will only apply to rows that are already loaded on the page, filtering has no impact on query parameters
  • Use quotes to match a longer phrase which contains spaces "mtor c1483f"

Sorting

  • Generally, the default sort order for tables is set to be first column ascending, however, specific tables may set a different default sort order.
  • Click on any column header arrows to sort by that column
  • Hold down the Shift key and click multiple columns to sort by more than one column, be sure to set ascending or descending order for a given column, before moving on to the next column.

Therapy Name Drugs Efficacy Evidence Clinical Trials
Abiraterone + Prednisone + Relugolix Abiraterone Prednisone Relugolix 0 1
Abiraterone + Relugolix Abiraterone Relugolix 0 1
Darolutamide + Relugolix Darolutamide Relugolix 0 1
Docetaxel + Relugolix Docetaxel Relugolix 0 1
Enzalutamide + Relugolix Enzalutamide Relugolix 0 1
Estradiol + Norethindrone + Relugolix Estradiol Norethindrone Relugolix 0 0
Relugolix Relugolix 0 3


Additional content available in CKB BOOST