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| Drug Name | Alpelisib |
| Trade Name | Piqray |
| Synonyms | BYL719 |
| Drug Descriptions |
Piqray (alpelisib) is a selective PIK3CA inhibitor that blocks activation of the PI3K signaling pathway and inhibits tumor growth (PMID: 23726034). Piqray (alpelisib) is FDA approved in combination with fulvestrant for use in postmenopausal women, and men, with advanced or metastatic hormone receptor (HR)-positive, ERBB2 (HER2)-negative, PIK3CA-mutant breast cancer (FDA.gov). |
| DrugClasses | PIK3CA inhibitor 23 |
| CAS Registry Number | 1217486-61-7 |
| NCIT ID | C94214 |
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