Drug Detail


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Drug Name Bicalutamide
Trade Name Casodex
Drug Descriptions

Casodex (bicalutamide) is an androgen-receptor antagonist that binds androgen receptors and inhibits androgen binding, therefore inhibits AR-dependent growth of tumor cells (PMID: 9428389). Casodex (bicalutamide) is approved, in combination with a luteinizing hormone-releasing hormone (LHRH) analog, for metastatic carcinoma of the prostate (FDA.gov).

DrugClasses Hormone - Anti-androgens 27


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Therapy Name Drugs Efficacy Evidence Clinical Trials
AT-101 + Bicalutamide AT-101 Bicalutamide 1 0
Bicalutamide Bicalutamide 1 19
Bicalutamide + Degarelix + Docetaxel Bicalutamide Degarelix Docetaxel 0 1
Bicalutamide + Docetaxel + Flutamide + Goserelin + Leuprolide + Nilutamide Bicalutamide Docetaxel Flutamide Goserelin Leuprolide Nilutamide 0 1
Bicalutamide + Docetaxel + Leuprolide Bicalutamide Docetaxel Leuprolide 0 2
Bicalutamide + Everolimus Bicalutamide Everolimus 1 0
Bicalutamide + Flutamide + Goserelin + Leuprolide + Nilutamide Bicalutamide Flutamide Goserelin Leuprolide Nilutamide 0 1
Bicalutamide + Gonadorelin Bicalutamide Gonadorelin 0 1
Bicalutamide + HSV-Tk + Leuprolide + Valacyclovir Bicalutamide HSV-Tk Leuprolide Valacyclovir 0 1
Bicalutamide + Ipilimumab + Nivolumab Bicalutamide Ipilimumab Nivolumab 0 1
Bicalutamide + Palbociclib Bicalutamide Palbociclib 0 1
Bicalutamide + Radium Ra 223 dichloride Bicalutamide Radium Ra 223 dichloride 0 1
Bicalutamide + Raloxifene Bicalutamide Raloxifene 0 1
Bicalutamide + Ribociclib Bicalutamide Ribociclib 0 1

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