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Drug Name Bicalutamide
Trade Name Casodex
Synonyms
Drug Descriptions

Casodex (bicalutamide) is an androgen-receptor antagonist that binds androgen receptors and inhibits androgen binding, therefore inhibits AR-dependent growth of tumor cells (PMID: 9428389). Casodex (bicalutamide) is approved, in combination with a luteinizing hormone-releasing hormone (LHRH) analog, for metastatic carcinoma of the prostate (FDA.gov).

DrugClasses Hormone - Anti-androgens 48
CAS Registry Number 90357-06-5
NCIT ID C1599

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Therapy Name Drugs Efficacy Evidence Clinical Trials
Abemaciclib + Bicalutamide Abemaciclib Bicalutamide 0 2
Abiraterone + Bicalutamide + Leuprolide + Prednisone + Talazoparib Abiraterone Bicalutamide Leuprolide Prednisone Talazoparib 0 1
Alpelisib + Bicalutamide Alpelisib Bicalutamide 0 0
AT-101 + Bicalutamide AT-101 Bicalutamide 0 0
Bicalutamide Bicalutamide 0 25
Bicalutamide + Buserelin Bicalutamide Buserelin 0 1
Bicalutamide + Darolutamide Bicalutamide Darolutamide 0 0
Bicalutamide + Degarelix Bicalutamide Degarelix 0 1
Bicalutamide + Degarelix + Docetaxel Bicalutamide Degarelix Docetaxel 0 1
Bicalutamide + Docetaxel + Flutamide + Goserelin + Leuprolide + Nilutamide Bicalutamide Docetaxel Flutamide Goserelin Leuprolide Nilutamide 0 1
Bicalutamide + Docetaxel + Leuprolide Bicalutamide Docetaxel Leuprolide 0 2
Bicalutamide + Dutasteride + Goserelin Bicalutamide Dutasteride Goserelin 0 1
Bicalutamide + Everolimus Bicalutamide Everolimus 0 0
Bicalutamide + Flutamide + Goserelin + Leuprolide + Nilutamide Bicalutamide Flutamide Goserelin Leuprolide Nilutamide 0 1
Bicalutamide + Gonadorelin Bicalutamide Gonadorelin 0 1
Bicalutamide + Goserelin Bicalutamide Goserelin 0 3
Bicalutamide + Histrelin acetate Bicalutamide Histrelin acetate 0 1
Bicalutamide + HSV-Tk + Leuprolide + Valacyclovir Bicalutamide HSV-Tk Leuprolide Valacyclovir 0 1
Bicalutamide + Ipilimumab + Nivolumab Bicalutamide Ipilimumab Nivolumab 0 1
Bicalutamide + Leuprolide Bicalutamide Leuprolide 0 3
Bicalutamide + Palbociclib Bicalutamide Palbociclib 0 1
Bicalutamide + Pyrotinib Bicalutamide Pyrotinib 0 0
Bicalutamide + Radium Ra 223 dichloride Bicalutamide Radium Ra 223 dichloride 0 1
Bicalutamide + Raloxifene Bicalutamide Raloxifene 0 1
Bicalutamide + Ribociclib Bicalutamide Ribociclib 0 1
Bicalutamide + Triptorelin Bicalutamide Triptorelin 0 4


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