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Drug Name | RMC-4550 |
Trade Name | |
Synonyms | RMC4550|RMC 4550 |
Drug Descriptions |
RMC-4550 is a small molecule allosteric inhibitor of Shp2 that blocks Ras-Raf-Mek-Erk pathway signaling, leading to tumor growth inhibition (PMID: 30104724). |
DrugClasses | SHP2 Inhibitor 19 |
CAS Registry Number | 2172651-73-7 |
NCIT ID | NA |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
Adagrasib + RMC-4550 | Adagrasib RMC-4550 | 0 | 0 |
Alectinib + RMC-4550 | Alectinib RMC-4550 | 1 | 0 |
Alpelisib + RMC-4550 + Sotorasib | Alpelisib RMC-4550 Sotorasib | 0 | 0 |
AZD4625 + RMC-4550 | AZD4625 RMC-4550 | 0 | 0 |
BAY-293 + Osimertinib + RMC-4550 | BAY-293 Osimertinib RMC-4550 | 0 | 0 |
BAY-293 + RMC-4550 | BAY-293 RMC-4550 | 0 | 0 |
Crizotinib + RMC-4550 | Crizotinib RMC-4550 | 0 | 0 |
D-1553 + RMC-4550 | D-1553 RMC-4550 | 0 | 0 |
Ipatasertib + RMC-4550 + Sotorasib | Ipatasertib RMC-4550 Sotorasib | 0 | 0 |
LY3214996 + RMC-4550 | LY3214996 RMC-4550 | 0 | 0 |
Osimertinib + RMC-4550 | Osimertinib RMC-4550 | 0 | 0 |
Pictilisib + RMC-4550 + Sotorasib | Pictilisib RMC-4550 Sotorasib | 0 | 0 |
RMC-4550 | RMC-4550 | 8 | 0 |
RMC-4550 + Sotorasib | RMC-4550 Sotorasib | 0 | 0 |