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Drug Name | AZD4547 |
Trade Name | |
Synonyms | AZD-4547 |
Drug Descriptions |
AZD4547 selectively binds and inhibits FGFR1, 2, and 3, which may result in the inhibition of FGFR-mediated signal transduction pathways and inhibition of tumor cell proliferation (PMID: 22369928, PMID: 30115694, PMID: 32463741). |
DrugClasses | FGFR1 Inhibitor 23 FGFR2 Inhibitor 16 FGFR3 Inhibitor 12 |
CAS Registry Number | 1035270-39-3 |
NCIT ID | C88272 |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
ABT-737 + AZD4547 | ABT-737 AZD4547 | 3 | 0 |
AZD4547 | AZD4547 | 80 | 3 |
AZD4547 + AZD8055 | AZD4547 AZD8055 | 2 | 0 |
AZD4547 + Buparlisib | AZD4547 Buparlisib | 4 | 0 |
AZD4547 + Capivasertib | AZD4547 Capivasertib | 1 | 0 |
AZD4547 + Cisplatin + Gemcitabine | AZD4547 Cisplatin Gemcitabine | 1 | 0 |
AZD4547 + Crizotinib | AZD4547 Crizotinib | 0 | 0 |
AZD4547 + Durvalumab | AZD4547 Durvalumab | 0 | 1 |
AZD4547 + Gefitinib | AZD4547 Gefitinib | 0 | 0 |
AZD4547 + Lapatinib | AZD4547 Lapatinib | 1 | 0 |
AZD4547 + Sapanisertib | AZD4547 Sapanisertib | 2 | 0 |
AZD4547 + Sirolimus | AZD4547 Sirolimus | 2 | 0 |
AZD4547 + Trametinib | AZD4547 Trametinib | 0 | 0 |
AZD4547 + Vistusertib | AZD4547 Vistusertib | 3 | 0 |