Drug Detail


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Drug Name 177Lu-PSMA-617
Trade Name
Synonyms Lu177-PSMA-617|Vipivotide tetraxetan Lu-177
Drug Descriptions

177Lu-PSMA-617 is a radioconjugate comprising a PSMA inhibitor radiolabeled with Lu177, which targets PSMA expressing cells, potentially resulting in decreased tumor growth (PMID: 25883127, PMID: 26795286, PMID: 32823294, PMID: 32760622).

CAS Registry Number 1703749-62-5
NCIT ID C148145


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Therapy Name Drugs Efficacy Evidence Clinical Trials
177Lu-J591 + 177Lu-PSMA-617 177Lu-J591 177Lu-PSMA-617 0 1
177Lu-PSMA-617 177Lu-PSMA-617 0 5
177Lu-PSMA-617 + Abemaciclib 177Lu-PSMA-617 Abemaciclib 0 1
177Lu-PSMA-617 + Pembrolizumab 177Lu-PSMA-617 Pembrolizumab 0 1

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