Drug Detail


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Drug Name Saracatinib
Trade Name
Synonyms AZD0530
Drug Descriptions

Saracatinib (AZD0530) is a multi-kinase inhibitor with activity against ABL and SRC, which may block proliferation, metastasis, and survival in cancer cells (PMID: 19393585, PMID: 32398945).

DrugClasses BCR-ABL Inhibitor 32 SRC Inhibitor 31
CAS Registry Number 379231-04-6
NCIT ID C48378


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Therapy Name Drugs Efficacy Evidence Clinical Trials
Afatinib + Saracatinib Afatinib Saracatinib 0 0
Cediranib + Saracatinib Cediranib Saracatinib 2 0
Ceritinib + Saracatinib Ceritinib Saracatinib 1 0
Dasatinib + Saracatinib Dasatinib Saracatinib 0 0
Docetaxel + Saracatinib Docetaxel Saracatinib 0 0
Enzalutamide + Saracatinib Enzalutamide Saracatinib 0 0
Gefitinib + PLX4720 + Saracatinib Gefitinib PLX4720 Saracatinib 1 0
Lapatinib + Saracatinib Lapatinib Saracatinib 0 0
Lorlatinib + Saracatinib Lorlatinib Saracatinib 2 0
Nilotinib + Saracatinib Nilotinib Saracatinib 0 0
Osimertinib + PF-573228 + Saracatinib Osimertinib PF-573228 Saracatinib 0 0
Osimertinib + Saracatinib Osimertinib Saracatinib 0 0
Ponatinib + Saracatinib Ponatinib Saracatinib 0 0
Saracatinib Saracatinib 3 1
Saracatinib + SCH772984 SCH772984 Saracatinib 0 0
Saracatinib + Selumetinib Saracatinib Selumetinib 0 0
Saracatinib + TAK-632 Saracatinib TAK-632 0 0
Saracatinib + Vemurafenib Saracatinib Vemurafenib 1 0

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