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Drug Name BMS-777607
Trade Name
Synonyms ASLAN002
Drug Descriptions

BMS-777607 (ASLAN002) is a small molecule that inhibits MET, MST1R (RON), TYRO3, and AXL, resulting in decreased downstream pathway activation, potentially resulting in decreased tumor cell growth and metastasis (PMID: 19260711, PMID: 20515943, PMID: 24233399, PMID: 26555154).

DrugClasses AXL Inhibitor 28 MET Inhibitor 56 RON Inhibitor 11 TYRO3 Inhibitor 8
CAS Registry Number 1025720-94-8
NCIT ID C74060

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Therapy Name Drugs Efficacy Evidence Clinical Trials
BMS-777607 BMS-777607 0 0
BMS-777607 + Buparlisib BMS-777607 Buparlisib 0 0
BMS-777607 + Trametinib BMS-777607 Trametinib 0 0


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